SCHEMBL8524665

SCHEMBL8524665

Cc1ccnc2c(S(=O)(=O)Nc3ccc4c(C(=O)NCc5ccc(C#N)cc5)cccc4c3)cccc12

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
PKLR P30613 3/20 0.40
POLB P06746 1/20 0.40
GRM4 Q14833 1/20 0.38
MCL1 Q07820 1/20 0.38
KLKB1 P03952 1/20 0.38
KLK1 P06870 1/20 0.38
CNR2 P34972 2/20 0.38
IMPDH2 P12268 1/20 0.38
ROCK1 Q13464 1/20 0.38
CTNNB1 P35222 1/20 0.37
TCF7L2 Q9NQB0 1/20 0.37
ALDH1A1 P00352 2/20 0.37
EGLN1 Q9GZT9 1/20 0.37
LMNA P02545 1/20 0.37
AKR1B1 P15121 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8525044 0.90 PKLR (0.49) MEN1KMT2APKLRALDH1A1EGLN1
SCHEMBL8524542 0.87 F2 (0.49) MEN1KMT2AKLKB1ALDH1A1
SCHEMBL8524454 0.84 PKLR (0.49) MEN1KMT2APKLRALDH1A1EGLN1
SCHEMBL8525447 0.84 PKLR (0.44) PKLRMCL1CNR2
SCHEMBL1110102 0.78 TUBB (0.46) MCL1KLKB1KLK1CNR2AKR1B1
SCHEMBL7358688 0.78 PKLR (0.47) MEN1KMT2APKLRALDH1A1EGLN1
Hydrochloric Acid SCHEMBL8525302 0.77 F2 (0.56) MEN1KMT2APKLRALDH1A1
SCHEMBL8525757 0.77 KMT2A (0.44) MEN1KMT2APKLRALDH1A1EGLN1
SCHEMBL8525059 0.75 HDAC2 (0.46) KLKB1KLK1CNR2IMPDH2CTNNB1
SCHEMBL8525755 0.73 HSP90AA1 (0.49) MCL1CNR2AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999029670-A2 AMINOCARBONYLTETRALIN AND DIHYDRONAPHTALENE DERIVATES AS THROMBIN INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-17 WO disclosed