SCHEMBL8524765

SCHEMBL8524765

CC(CC(=O)O)c1cccc(CCNC(=O)c2cccc(Nc3nc4ccccc4[nH]3)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.54
ITGB3 P05106 5/20 0.53
ITGAV P06756 5/20 0.53
HTT P42858 3/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45
MMP8 P22894 1/20 0.45
LMNA P02545 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
MAPT P10636 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
AURKB Q96GD4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7863185 0.92 AKR1C3 (0.56) AKR1C3ITGB3ITGAVHTTNPC1
SCHEMBL8525720 0.89 HDAC11 (0.44) AKR1C3ITGB3ITGAVNPC1RAB9A
SCHEMBL8524766 0.84 AKR1C3 (0.58) AKR1C3ITGB3ITGAVHTTNPC1
SCHEMBL8526841 0.82 AKR1C3 (0.54) AKR1C3ITGB3ITGAVHTTNPC1
SCHEMBL7863112 0.81 ROCK1 (0.47) AKR1C3ITGB3ITGAVHTTNPC1
SCHEMBL8534047 0.80 AKR1C3 (0.57) AKR1C3ITGB3ITGAVHTTNPC1
SCHEMBL8524575 0.77 LMNA (0.42) ITGB3ITGAVNPC1RAB9ASMN1; SMN2
SCHEMBL8525722 0.74 HDAC11 (0.46) AKR1C3ITGB3ITGAVNPC1RAB9A
SCHEMBL13002087 0.73 AKR1C3 (0.73) AKR1C3ITGB3ITGAVHTTNPC1
SCHEMBL29624703 0.72 AKR1C3 (0.77) AKR1C3HTTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed