SCHEMBL8526841

SCHEMBL8526841

CCC(CC(=O)O)c1cccc(CNC(=O)c2cccc(Nc3nc4ccccc4[nH]3)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.54
ITGB3 P05106 4/20 0.49
ITGAV P06756 4/20 0.49
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
HTT P42858 3/20 0.46
MAPT P10636 2/20 0.46
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
HDAC6 Q9UBN7 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
LMNA P02545 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
HDAC11 Q96DB2 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7863185 0.90 AKR1C3 (0.56) AKR1C3ITGB3ITGAVMEN1KMT2A
SCHEMBL8526505 0.89 ROCK1 (0.46) AKR1C3MEN1KMT2AHTTMAPT
SCHEMBL8524765 0.82 AKR1C3 (0.54) AKR1C3ITGB3ITGAVMEN1KMT2A
SCHEMBL7863112 0.79 ROCK1 (0.47) AKR1C3ITGB3ITGAVMEN1KMT2A
SCHEMBL8534047 0.79 AKR1C3 (0.57) AKR1C3ITGB3ITGAVMEN1KMT2A
SCHEMBL7862019 0.76 LMNA (0.45) ITGB3HTTMAPTALDH1A1LMNA
SCHEMBL8524766 0.76 AKR1C3 (0.58) AKR1C3ITGB3ITGAVMEN1KMT2A
SCHEMBL7864751 0.75 SIRT2 (0.41) ITGB3ITGAVHTTALDH1A1GAA
SCHEMBL22703577 0.73 AKR1C3 (0.73) AKR1C3MEN1KMT2AHDAC6LMNA
SCHEMBL29624703 0.72 AKR1C3 (0.77) AKR1C3MEN1KMT2AHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed