SCHEMBL8525722

SCHEMBL8525722

COc1ccc2[nH]c(Nc3cccc(C(=O)NC(C)c4cccc(C(C)CC(=O)O)c4)c3)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC11 Q96DB2 2/20 0.46
ITGB3 P05106 1/20 0.44
ITGAV P06756 1/20 0.44
AKR1C3 P42330 1/20 0.43
NPC1 O15118 1/20 0.43
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ROCK2 O75116 10/20 0.43
ROCK1 Q13464 5/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GPR139 Q6DWJ6 3/20 0.42
BACE1 P56817 1/20 0.41
BACE2 Q9Y5Z0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8524766 0.88 AKR1C3 (0.58) HDAC11ITGB3ITGAVAKR1C3NPC1
SCHEMBL7863112 0.87 ROCK1 (0.47) HDAC11ITGB3ITGAVAKR1C3NPC1
SCHEMBL8525720 0.86 HDAC11 (0.44) HDAC11ITGB3ITGAVAKR1C3NPC1
SCHEMBL8534053 0.81 HDAC11 (0.45) HDAC11ITGB3ITGAVAKR1C3NPC1
SCHEMBL8526505 0.78 ROCK1 (0.46) HDAC11AKR1C3NPC1PKMRAB9A
SCHEMBL7863185 0.75 AKR1C3 (0.56) HDAC11ITGB3ITGAVAKR1C3NPC1
SCHEMBL8524765 0.74 AKR1C3 (0.54) HDAC11ITGB3ITGAVAKR1C3NPC1
SCHEMBL8524582 0.72 ROCK2 (0.40) ITGB3ITGAVROCK2ROCK1
SCHEMBL8534047 0.69 AKR1C3 (0.57) HDAC11ITGB3ITGAVAKR1C3NPC1
SCHEMBL3786660 0.69 KMT2A (0.56) HDAC11AKR1C3NPC1PKMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed