SCHEMBL7863112

SCHEMBL7863112

COc1ccc2[nH]c(Nc3cccc(C(=O)NCc4cccc(C(C)CC(=O)O)c4)c3)nc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.47
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
ALDH1A1 P00352 2/20 0.45
GAA P10253 2/20 0.45
USP2 O75604 1/20 0.45
HDAC11 Q96DB2 2/20 0.45
MMP13 P45452 3/20 0.45
ROCK2 O75116 2/20 0.44
ITGB3 P05106 2/20 0.43
ITGAV P06756 2/20 0.43
HPGDS O60760 1/20 0.43
PRKCA P17252 1/20 0.42
GRK2 P25098 1/20 0.42
AKR1C3 P42330 1/20 0.42
MAPT P10636 2/20 0.42
HTT P42858 1/20 0.42
NPC1 O15118 1/20 0.42
PKM P14618 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8525720 0.92 HDAC11 (0.44) ROCK1MEN1KMT2AALDH1A1HDAC11
SCHEMBL8526505 0.91 ROCK1 (0.46) ROCK1MEN1KMT2AALDH1A1GAA
SCHEMBL7863185 0.89 AKR1C3 (0.56) MEN1KMT2AALDH1A1GAAHDAC11
SCHEMBL8525722 0.87 HDAC11 (0.46) ROCK1HDAC11ROCK2ITGB3ITGAV
SCHEMBL8534053 0.86 HDAC11 (0.45) ROCK1MEN1KMT2AALDH1A1GAA
SCHEMBL8524765 0.81 AKR1C3 (0.54) MEN1KMT2AALDH1A1GAAHDAC11
SCHEMBL8526841 0.79 AKR1C3 (0.54) MEN1KMT2AALDH1A1GAAHDAC11
SCHEMBL8524766 0.75 AKR1C3 (0.58) MEN1KMT2AALDH1A1HDAC11ITGB3
SCHEMBL8534047 0.74 AKR1C3 (0.57) MEN1KMT2AALDH1A1GAAHDAC11
SCHEMBL7861566 0.73 ROCK2 (0.41) ROCK1ROCK2ITGB3ITGAVPRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed