SCHEMBL8534053

SCHEMBL8534053

COc1ccc2[nH]c(Nc3cccc(C(=O)NCc4ccccc4C(C)CC(=O)O)c3)nc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC11 Q96DB2 3/20 0.45
AKR1C3 P42330 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 1/20 0.44
PKM P14618 1/20 0.44
RAB9A P51151 1/20 0.44
GAA P10253 3/20 0.42
HPGD P15428 1/20 0.42
MAPT P10636 4/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
ALDH1A1 P00352 2/20 0.42
HTT P42858 1/20 0.42
EPHX2 P34913 2/20 0.41
BCHE P06276 1/20 0.41
ROCK1 Q13464 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8534047 0.89 AKR1C3 (0.57) HDAC11AKR1C3SMN1; SMN2NPC1PKM
SCHEMBL7863112 0.86 ROCK1 (0.47) HDAC11AKR1C3SMN1; SMN2NPC1PKM
SCHEMBL8525720 0.81 HDAC11 (0.44) HDAC11AKR1C3SMN1; SMN2NPC1PKM
SCHEMBL8525722 0.81 HDAC11 (0.46) HDAC11AKR1C3SMN1; SMN2NPC1PKM
SCHEMBL8526505 0.80 ROCK1 (0.46) HDAC11AKR1C3SMN1; SMN2NPC1PKM
SCHEMBL7863185 0.76 AKR1C3 (0.56) HDAC11AKR1C3SMN1; SMN2NPC1RAB9A
SCHEMBL8524765 0.71 AKR1C3 (0.54) HDAC11AKR1C3SMN1; SMN2NPC1RAB9A
SCHEMBL8524766 0.70 AKR1C3 (0.58) HDAC11AKR1C3SMN1; SMN2NPC1PKM
SCHEMBL8526841 0.69 AKR1C3 (0.54) HDAC11AKR1C3SMN1; SMN2NPC1PKM
SCHEMBL11703469 0.69 RAB9A (0.73) SMN1; SMN2NPC1PKMRAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773646-A INTEGRIN INHIBITORS G. D. SEARLE & CO. (US) 1998-06-30 US disclosed