SCHEMBL8526169

SCHEMBL8526169

CCOC(=O)CNC(=O)NCc1ccccc1C#N

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPID Q08752 5/20 0.61
PPIB P23284 1/20 0.52
PPIA P62937 1/20 0.52
PPIG Q13427 1/20 0.52
NLRP3 Q96P20 2/20 0.49
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MAPT P10636 1/20 0.45
P2RX7 Q99572 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.43
HTT P42858 1/20 0.43
AVPR2 P30518 1/20 0.43
POLB P06746 1/20 0.41
TSHR P16473 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5449507 0.80 PPID (0.66) PPIDPPIBPPIAPPIGNLRP3
SCHEMBL2053656 0.78 PPID (0.67) PPIDPPIBPPIAPPIGALDH1A1
SCHEMBL7219075 0.78 NLRP3 (0.55) NLRP3ALDH1A1KDM4EGAAL3MBTL1
SCHEMBL10065403 0.78 P2RX7 (0.49) ALDH1A1KDM4EGAAP2RX7POLB
SCHEMBL12643825 0.76 PPID (1.00) PPIDPPIBPPIAPPIGALDH1A1
SCHEMBL8138307 0.76 PPID (0.69) PPIDPPIBPPIAPPIGALDH1A1
SCHEMBL6925202 0.76 P2RX7 (0.49) ALDH1A1KDM4EGAAL3MBTL1P2RX7
SCHEMBL15832182 0.75 PPID (0.67) PPIDPPIBPPIAPPIGNLRP3
SCHEMBL26661046 0.75 CYP4F2 (0.63) NLRP3ALDH1A1KDM4EGAAL3MBTL1
SCHEMBL31036963 0.75 P2RX7 (0.55) ALDH1A1GAAL3MBTL1P2RX7HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed