SCHEMBL8526111

SCHEMBL8526111

CCCCc1ccc(C(=O)N(Cc2ccc(CNC(N)=O)cc2)[C@H](CCCNC(=N)N)C(=O)NCC(=O)O)cc1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
CTSK P43235 1/20 0.37
SPHK1 Q9NYA1 1/20 0.37
ST14 Q9Y5Y6 1/20 0.36
OPRK1 P41145 1/20 0.36
ITGB3 P05106 2/20 0.35
ITGA2B P08514 2/20 0.35
MASP2 O00187 1/20 0.34
F2 P00734 1/20 0.34
PPARG P37231 1/20 0.34
S1PR2 O95136 1/20 0.33
S1PR4 O95977 1/20 0.33
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
PROC P04070 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8526313 0.91 TMEM97 (0.41) TMEM97SIGMAR1CTSKSPHK1ST14
SCHEMBL8528194 0.84 F7 (0.40) TMEM97SIGMAR1F2PPARGPROC
SCHEMBL8526482 0.83 KMT2A (0.40) ITGB3ITGA2BF2PROC
SCHEMBL8528338 0.82 CCR2 (0.36) F2
SCHEMBL8527067 0.79 ALDH1A1 (0.41) TMEM97SIGMAR1OPRK1
SCHEMBL7039253 0.77 CASR (0.38) ITGB3ITGA2B
SCHEMBL8526200 0.77 HDAC1 (0.35)
SCHEMBL8121122 0.76 TMEM97 (0.42) TMEM97SIGMAR1CTSKOPRK1ITGB3
SCHEMBL7045274 0.76 KDM4E (0.42) ITGB3
SCHEMBL8122129 0.75 F7 (0.40) TMEM97SIGMAR1F2PPARGPROC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed