SCHEMBL8527872

SCHEMBL8527872

COc1ccc(OC)c2c1COC(C(=O)CBr)C2

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 3/20 0.40
CYP1A2 P05177 1/20 0.40
HPGDS O60760 1/20 0.35
ACHE P22303 1/20 0.35
ALDH1A1 P00352 3/20 0.33
MTNR1A P48039 2/20 0.33
MTNR1B P49286 2/20 0.33
HPGD P15428 2/20 0.33
MIF P14174 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530160 0.83 ADRA1A (0.38) ADRA1ACYP1A2ACHEALDH1A1MTNR1A
SCHEMBL8529815 0.83 ADRA1A (0.46) ADRA1ACYP1A2ACHEALDH1A1MTNR1A
SCHEMBL8527137 0.82 MIF (0.45) ADRA1ACYP1A2ACHEALDH1A1MTNR1A
SCHEMBL8527470 0.82 CYP1A2 (0.47) ADRA1ACYP1A2ACHEALDH1A1MTNR1A
SCHEMBL8901669 0.81 ADRA1A (0.36) ADRA1ACYP1A2ACHEALDH1A1MTNR1A
SCHEMBL8527142 0.81 MIF (0.46) ADRA1ACYP1A2ACHEALDH1A1MTNR1A
SCHEMBL8901644 0.79 CTDSP1 (0.44) ADRA1ACYP1A2ALDH1A1HPGD
SCHEMBL8531328 0.78 ADRA1A (0.41) ADRA1ACYP1A2ACHEALDH1A1MTNR1A
SCHEMBL8533392 0.77 ADRA1A (0.42) ADRA1ACYP1A2ACHEALDH1A1MTNR1A
SCHEMBL8527222 0.76 ADRA1A (0.39) ADRA1ACYP1A2ACHEALDH1A1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5606037-A Processes antineoplastic heteronaphthoquinones BIOCHEM PHARMA INC. (CA) 1997-02-25 US claimed
US-5736523-A ADMINISTERING TO THE MAMMAL SUFFERING FROM CANCER BIOCHEM PHARMA INC. (CA) 1998-04-07 US disclosed
US-5606037-A Processes antineoplastic heteronaphthoquinones BIOCHEM PHARMA INC. (CA) 1997-02-25 US disclosed
EP-0659190-A1 ANTINEOPLASTIC HETERONAPHTHOQUINONES BIOCHEM PHARMA INC (CA) 1995-06-28 EP disclosed
WO-1994011382-A1 ANTINEOPLASTIC HETERONAPHTHOQUINONES BIOCHEM PHARMA INC. (CA) 1994-05-26 WO disclosed