SCHEMBL8528642

SCHEMBL8528642

[CH2]c1cn(CC(=O)OCC)c2ccccc12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.67
MAPT P10636 2/20 0.66
LMNA P02545 1/20 0.66
POLB P06746 1/20 0.64
L3MBTL1 Q9Y468 1/20 0.64
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
MEN1 O00255 1/20 0.59
CRHBP P24387 1/20 0.59
KMT2A Q03164 1/20 0.59
CRHR2 Q13324 1/20 0.59
TSHR P16473 3/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
CREBBP Q92793 1/20 0.52
KDM4E B2RXH2 3/20 0.52
RAB9A P51151 1/20 0.51
HPGD P15428 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8528645 0.85 ALDH1A1 (0.71) ALDH1A1MAPTLMNAPOLBL3MBTL1
SCHEMBL8531842 0.85 GAA (0.68) ALDH1A1MAPTLMNAPOLBL3MBTL1
SCHEMBL13490809 0.84 ALDH1A1 (0.69) ALDH1A1MAPTLMNAPOLBL3MBTL1
SCHEMBL8527333 0.83 L3MBTL1 (0.52) ALDH1A1MAPTLMNAPOLBL3MBTL1
SCHEMBL14880155 0.83 ALDH1A1 (0.67) ALDH1A1MAPTLMNAPOLBL3MBTL1
SCHEMBL8530927 0.82 GAA (0.49) ALDH1A1MAPTLMNAPOLBL3MBTL1
SCHEMBL28623979 0.82 LMNA (0.76) ALDH1A1MAPTLMNAPOLBL3MBTL1
Hydrochloric Acid SCHEMBL14876437 0.82 ALDH1A1 (0.66) ALDH1A1MAPTLMNAPOLBL3MBTL1
SCHEMBL18171795 0.82 ALDH1A1 (0.66) ALDH1A1MAPTLMNAPOLBL3MBTL1
SCHEMBL1250151 0.81 ALDH1A1 (1.00) ALDH1A1MAPTLMNAPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0460679-B1 Endothelin antagonistic peptide derivatives BANYU PHARMA CO LTD (JP) 1998-10-28 EP disclosed
US-5691315-A CARDIOVASCULAR DISORDERS; VASODILATOR; BRONCHODILATOR BANYU PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
US-5470833-A Vasodilators, bronchodilators BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-11-28 US disclosed
US-5444152-A Vasolidator or bronchodilator BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-08-22 US disclosed
EP-0460679-A2 Endothelin antagonistic peptide derivatives Banyu Pharmaceutical Co., Ltd. (JP) 1991-12-11 EP disclosed