SCHEMBL8528882

SCHEMBL8528882

COc1nc(N)nc2c1ncn2[C@@H]1O[C@H](CO[Si](C)(C)C(C)(C)C)[C@@H](O)[C@@H]1O[Si](C)(C)C(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HINT1 P49773 2/20 0.45
NT5E P21589 2/20 0.45
ADORA3 P0DMS8 3/20 0.44
CYP2C19 P33261 1/20 0.43
ADORA1 P30542 3/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42
SLC29A1 Q99808 5/20 0.40
RNASEL Q05823 1/20 0.40
PGK1 P00558 1/20 0.39
PGK2 P07205 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8529223 0.93 HINT1 (0.45) HINT1NT5EADORA3CYP2C19ADORA1
SCHEMBL8533343 0.92 HINT1 (0.40) HINT1NT5EADORA3CYP2C19ADORA1
SCHEMBL8534590 0.91 HINT1 (0.54) HINT1NT5EADORA3CYP2C19ADORA1
SCHEMBL8529436 0.87 ALDH1A1 (0.48) HINT1NT5EADORA3CYP2C19ADORA1
SCHEMBL8533171 0.87 HINT1 (0.40) HINT1NT5EADORA3CYP2C19ADORA1
SCHEMBL8529887 0.87 HINT1 (0.40) HINT1NT5EADORA3CYP2C19ADORA1
SCHEMBL8529066 0.85 CYP2C19 (0.48) ADORA3CYP2C19ADORA1ADORA2AADORA2B
SCHEMBL8530373 0.85 ADORA2A (0.40) HINT1NT5ECYP2C19ADORA1ADORA2A
SCHEMBL8529155 0.84 ALDH1A1 (0.52) HINT1NT5EADORA3CYP2C19ADORA1
SCHEMBL8988189 0.84 HINT1 (0.38) HINT1NT5EADORA3CYP2C19ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821236-A Tumor treatment with arabinofuranosyl purine derivatives GLAXO WELLCOME INC. (US) 1998-10-13 US disclosed
US-5747472-A ANTICARCINOGENIC AGENTS AND ANTITUMOR AGENTS GLAXO WELLCOME INC. (US) 1998-05-05 US disclosed
US-5492897-A ANTITUMOR AGENTS, AUTOIMMUNE DISEASES BURROUGHS WELLCOME CO. (141) (US) 1996-02-20 US disclosed
US-5424295-A Useful in treatment of varicella-zoster virus infections BURROUGHS WELLCOME CO. (US) 1995-06-13 US disclosed
WO-1992001456-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-02-06 WO disclosed