SCHEMBL8533343

SCHEMBL8533343

COc1nc(N)nc2c1ncn2[C@@H]1O[C@H](CO[Si](C)(C)C(C)(C)C)[C@@H](O[Si](C)(C)C(C)(C)C)[C@@H]1O[Si](C)(C)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HINT1 P49773 2/20 0.40
NT5E P21589 2/20 0.39
CYP2C19 P33261 1/20 0.39
SLC29A1 Q99808 5/20 0.38
ADORA3 P0DMS8 3/20 0.38
ADORA1 P30542 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
PGK1 P00558 1/20 0.35
PGK2 P07205 1/20 0.35
HSP90B1 P14625 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8529223 0.92 HINT1 (0.45) HINT1NT5ECYP2C19SLC29A1ADORA3
SCHEMBL8528882 0.92 HINT1 (0.45) HINT1NT5ECYP2C19SLC29A1ADORA3
SCHEMBL8529436 0.92 ALDH1A1 (0.48) HINT1NT5ECYP2C19SLC29A1ADORA3
SCHEMBL8529887 0.91 HINT1 (0.40) HINT1NT5ECYP2C19SLC29A1ADORA3
SCHEMBL8530373 0.91 ADORA2A (0.40) HINT1NT5ECYP2C19SLC29A1ADORA1
SCHEMBL8533171 0.91 HINT1 (0.40) HINT1NT5ECYP2C19SLC29A1ADORA3
SCHEMBL8529066 0.90 CYP2C19 (0.48) CYP2C19SLC29A1ADORA3ADORA1ADORA2A
SCHEMBL8988189 0.88 HINT1 (0.38) HINT1NT5ECYP2C19SLC29A1ADORA3
SCHEMBL20635016 0.88 HINT1 (0.42) HINT1NT5ECYP2C19SLC29A1ADORA3
SCHEMBL8530537 0.87 P2RX3 (0.46) HINT1NT5ESLC29A1ADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821236-A Tumor treatment with arabinofuranosyl purine derivatives GLAXO WELLCOME INC. (US) 1998-10-13 US disclosed
US-5747472-A ANTICARCINOGENIC AGENTS AND ANTITUMOR AGENTS GLAXO WELLCOME INC. (US) 1998-05-05 US disclosed
US-5492897-A ANTITUMOR AGENTS, AUTOIMMUNE DISEASES BURROUGHS WELLCOME CO. (141) (US) 1996-02-20 US disclosed