SCHEMBL8529007

SCHEMBL8529007

COc1nc(N)nc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](OC(=O)c2ccccc2)[C@@H]1O

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 3/20 0.50
P2RY11 Q96G91 1/20 0.50
CYP2C19 P33261 1/20 0.49
ENPP1 P22413 1/20 0.49
ADORA2A P29274 6/20 0.49
ADORA2B P29275 5/20 0.49
ADORA3 P0DMS8 4/20 0.49
ADORA1 P30542 4/20 0.49
HINT1 P49773 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8529895 0.93 P2RY11 (0.54) SLC29A1P2RY11CYP2C19ADORA2AADORA2B
SCHEMBL17359509 0.85 P2RX3 (0.49) SLC29A1P2RY11CYP2C19ADORA2AADORA2B
SCHEMBL8529892 0.85 CYP2C19 (0.52) SLC29A1CYP2C19ADORA2AADORA2BADORA3
SCHEMBL17357579 0.82 P2RY11 (0.46) SLC29A1P2RY11CYP2C19ADORA2AADORA2B
SCHEMBL29479248 0.82 HINT1 (0.59) P2RY11ENPP1HINT1
Nelarabine SCHEMBL14031852 0.81 CYP2C19 (0.71) SLC29A1CYP2C19ADORA2AADORA2BADORA3
Nelarabine SCHEMBL18321891 0.81 CYP2C19 (0.71) SLC29A1CYP2C19ADORA2AADORA2BADORA3
Nelarabine SCHEMBL2143756 0.81 CYP2C19 (0.71) SLC29A1CYP2C19ADORA2AADORA2BADORA3
Nelarabine SCHEMBL20769831 0.81 CYP2C19 (0.71) SLC29A1CYP2C19ADORA2AADORA2BADORA3
Nelarabine SCHEMBL13657986 0.81 CYP2C19 (0.71) SLC29A1CYP2C19ADORA2AADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821236-A Tumor treatment with arabinofuranosyl purine derivatives GLAXO WELLCOME INC. (US) 1998-10-13 US disclosed
US-5747472-A ANTICARCINOGENIC AGENTS AND ANTITUMOR AGENTS GLAXO WELLCOME INC. (US) 1998-05-05 US disclosed
US-5492897-A ANTITUMOR AGENTS, AUTOIMMUNE DISEASES BURROUGHS WELLCOME CO. (141) (US) 1996-02-20 US disclosed
US-5424295-A Useful in treatment of varicella-zoster virus infections BURROUGHS WELLCOME CO. (US) 1995-06-13 US disclosed