SCHEMBL8529581

SCHEMBL8529581

COC(=O)Cc1cn(C)c2ccc(C(=O)O)cc12

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CPT1A P50416 2/20 0.49
CPT1B Q92523 2/20 0.49
CPT2 P23786 1/20 0.49
AKR1C3 P42330 1/20 0.49
KDM4E B2RXH2 3/20 0.46
NQO2 P16083 1/20 0.45
MTNR1A P48039 1/20 0.45
MTNR1B P49286 1/20 0.45
SPR P35270 1/20 0.44
ICMT O60725 1/20 0.43
HASPIN Q8TF76 1/20 0.43
S1PR2 O95136 1/20 0.42
F2 P00734 1/20 0.42
PRSS1 P07477 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2686872 0.83 SPR (0.62) AKR1C3KDM4ENQO2MTNR1AMTNR1B
SCHEMBL2686296 0.82 MTNR1A (0.65) AKR1C3NQO2MTNR1AMTNR1B
SCHEMBL20604920 0.82 KDM4E (0.47) AKR1C3KDM4ENQO2MTNR1AMTNR1B
SCHEMBL4012453 0.79 KDM4E (0.65) KDM4ES1PR2
SCHEMBL31498840 0.79 KDM4E (0.65) KDM4ES1PR2
SCHEMBL8536461 0.78 PLA2G4A (0.61) CPT1ACPT1BCPT2
SCHEMBL2807415 0.78 NR4A2 (0.46) CPT1ACPT1BCPT2KDM4E
SCHEMBL2804273 0.77 NR4A2 (0.45) KDM4E
SCHEMBL3352657 0.77 HPGD (0.49) CPT1ACPT1BCPT2KDM4ENQO2
SCHEMBL2804408 0.76 PLA2G4A (0.46) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0489547-B1 A process for the preparation of a 3-alkylated indole, intermediates, and a process for the preparation of a derivative thereof ZENECA LTD (GB) 1998-07-29 EP disclosed
US-5280125-A Chemical process for the preparation of 3-alkylated indole IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-01-18 US disclosed
EP-0489547-A1 A process for the preparation of a 3-alkylated indole, intermediates, and a process for the preparation of a derivative thereof ZENECA LIMITED (GB) 1992-06-10 EP disclosed