SCHEMBL8530758

SCHEMBL8530758

O=C(O)c1ccc(F)cc1Sc1cccc(F)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 5/20 0.45
DCLRE1B Q9H816 1/20 0.42
EPHX1 P07099 1/20 0.42
KEAP1 Q14145 1/20 0.42
NOTUM Q6P988 1/20 0.39
HAO1 Q9UJM8 1/20 0.39
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GRIK1 P39086 1/20 0.38
RHEB Q15382 1/20 0.38
CES2 O00748 2/20 0.38
CES1 P23141 2/20 0.38
POLB P06746 1/20 0.38
KDM4C Q9H3R0 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10597129 0.90 ALDH1A1 (0.47) SLC6A9KEAP1ALDH1A1GLAL3MBTL1
SCHEMBL11760302 0.88 GRIK1 (0.49) SLC6A9ALDH1A1GRIK1RHEB
SCHEMBL8533329 0.87 SLC6A9 (0.48) SLC6A9DCLRE1BEPHX1KEAP1NOTUM
SCHEMBL26676266 0.87 SIRT1 (0.51) SLC6A9EPHX1ALDH1A1GLAL3MBTL1
SCHEMBL8531521 0.86 SLC6A9 (0.42) SLC6A9EPHX1HAO1ALDH1A1CES2
SCHEMBL8533536 0.85 RHEB (0.47) SLC6A9KEAP1NOTUMALDH1A1GLA
SCHEMBL8529753 0.82 SLC6A9 (0.47) SLC6A9EPHX1ALDH1A1
SCHEMBL29269655 0.81 KDM4C (0.50) SLC6A9EPHX1HAO1ALDH1A1L3MBTL1
SCHEMBL30402222 0.81 KDM4C (0.50) SLC6A9EPHX1HAO1ALDH1A1L3MBTL1
SCHEMBL4442324 0.80 POLB (0.53) KEAP1ALDH1A1L3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0859757-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS Farmak A.S. (CZ) 1998-08-26 EP disclosed
WO-1997017325-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS FARMAK A.S. (CZ) 1997-05-15 WO disclosed