SCHEMBL8533222

SCHEMBL8533222

CC(C)Oc1ccc(-c2ccnc(N3CCC4(CCNCC4)C3)n2)cc1C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.38
ALDH1A1 P00352 5/20 0.38
HSD17B10 Q99714 5/20 0.38
CYP1A2 P05177 3/20 0.38
KMO O15229 1/20 0.37
CYP3A4 P08684 4/20 0.36
TSHR P16473 4/20 0.36
LRRK2 Q5S007 1/20 0.36
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
CDC42BPB Q9Y5S2 1/20 0.35
MAP3K12 Q12852 1/20 0.34
HPGD P15428 2/20 0.34
DYRK1A Q13627 2/20 0.34
MAPK14 Q16539 1/20 0.33
CCR4 P51679 1/20 0.33
S1PR1 P21453 1/20 0.33
CDK1 P06493 1/20 0.32
CDK4 P11802 1/20 0.32
CCNB1 P14635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8511790 0.87 ROCK2 (0.41) ALDH1A1KMOLRRK2ROCK2S1PR1
Hydrochloric Acid SCHEMBL8511580 0.86 ROCK2 (0.41) ALDH1A1KMOLRRK2ROCK2S1PR1
Hydrochloric Acid SCHEMBL8512525 0.86 ROCK2 (0.41) ALDH1A1KMOLRRK2ROCK2S1PR1
SCHEMBL8514660 0.84 KMO (0.38) CYP2D6ALDH1A1HSD17B10CYP1A2KMO
SCHEMBL8510230 0.84 KARS1 (0.34) LRRK2PIM1PIM3PIM2
SCHEMBL8510713 0.82 KMO (0.39) KMOLRRK2DKK1
SCHEMBL8510840 0.81 KMO (0.43) ALDH1A1HSD17B10CYP1A2KMOCYP3A4
SCHEMBL9612861 0.80 S1PR1 (0.41) KMOS1PR1DKK1
SCHEMBL8510739 0.79 ZAP70 (0.41) KMOLRRK2ROCK2ROCK1DKK1
SCHEMBL8510734 0.79 ZAP70 (0.41) KMOLRRK2ROCK2ROCK1DKK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed