SCHEMBL8510230

SCHEMBL8510230

CC(C)Oc1ccc(-c2ccnc(N3CCC4(CCNCC4)C3)n2)cc1C(C)(C)C.CC(C)c1cc(-c2cccc(N3CCNCC3)n2)ccc1OCC(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KARS1 Q15046 3/20 0.34
LRRK2 Q5S007 1/20 0.33
ITGB2 P05107 7/20 0.32
ICAM1 P05362 7/20 0.32
ITGAL P20701 7/20 0.32
PIM1 P11309 4/20 0.31
PIM3 Q86V86 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
TLR9 Q9NR96 1/20 0.31
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
ADRB1 P08588 1/20 0.31
PRKD1 Q15139 1/20 0.31
PRKD2 Q9BZL6 1/20 0.31
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8533222 0.84 CYP2D6 (0.38) LRRK2PIM1PIM3PIM2
SCHEMBL8515290 0.80 KARS1 (0.45) KARS1ITGB2ICAM1ITGALPIM1
Hydrochloric Acid SCHEMBL8512524 0.79 KARS1 (0.44) KARS1ITGB2ICAM1ITGALPIM1
SCHEMBL8514718 0.77 KARS1 (0.46) KARS1PIM1PIM3PIM2HTR2C
SCHEMBL8514744 0.77 S1PR1 (0.41) KARS1PIM1PIM3PIM2PRKD1
Hydrochloric Acid SCHEMBL8511433 0.76 KARS1 (0.45) KARS1PIM1PIM3PIM2HTR2C
Hydrochloric Acid SCHEMBL8512940 0.76 S1PR1 (0.41) KARS1PIM1PIM3PIM2PRKD1
SCHEMBL8511790 0.76 ROCK2 (0.41) LRRK2ADRB1PRKD1PRKD2
Hydrochloric Acid SCHEMBL8512525 0.76 ROCK2 (0.41) LRRK2ADRB1PRKD1PRKD2
Hydrochloric Acid SCHEMBL8511580 0.76 ROCK2 (0.41) LRRK2ADRB1PRKD1PRKD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed