SCHEMBL8533347

SCHEMBL8533347

COc1cc(Sc2ccccc2C(=O)N(C)C)ccc1F

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.50
ALDH1A1 P00352 2/20 0.50
MEN1 O00255 1/20 0.50
MAPT P10636 1/20 0.50
KMT2A Q03164 1/20 0.50
CXCR2 P25025 2/20 0.41
AR P10275 1/20 0.40
GAA P10253 1/20 0.40
SLC6A4 P31645 1/20 0.40
ITGAL P20701 1/20 0.40
GRM4 Q14833 1/20 0.39
SLC6A9 P48067 5/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6216437 0.86 NSD2 (0.44) HPGDALDH1A1ARITGALGRM4
SCHEMBL8533973 0.85 ALDH1A1 (0.60) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL5833804 0.78 KMT2A (0.50) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL11749787 0.75 SIRT1 (0.61) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL8534092 0.74 ALDH1A1 (0.69) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL8530163 0.74 ALDH1A1 (0.54) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL8529733 0.74 MEN1 (0.54) HPGDALDH1A1MEN1MAPTKMT2A
Hydrochloric Acid SCHEMBL8586417 0.73 SLC6A4 (0.57) ALDH1A1SLC6A4
SCHEMBL232284 0.73 HTT (0.50) HPGDALDH1A1MEN1KMT2AAR
SCHEMBL8533938 0.73 ALDH1A1 (0.53) HPGDALDH1A1MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0859757-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS Farmak A.S. (CZ) 1998-08-26 EP disclosed
WO-1997017325-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS FARMAK A.S. (CZ) 1997-05-15 WO disclosed