SCHEMBL8533973

SCHEMBL8533973

COc1cc(Sc2ccccc2C(=O)N(C)C)ccc1Cl

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.60
HPGD P15428 3/20 0.60
MAPT P10636 2/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
SLC6A4 P31645 1/20 0.47
HTT P42858 1/20 0.46
AR P10275 1/20 0.40
GAA P10253 1/20 0.40
GRM4 Q14833 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
SLC6A9 P48067 4/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530235 0.86 AR (0.43) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL8533409 0.86 CLCN2 (0.46) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL8533347 0.85 HPGD (0.50) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL5833804 0.78 KMT2A (0.50) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL11480340 0.75 MMP2 (0.60) HPGDSLC6A4ARGRM4HDAC6
SCHEMBL11749787 0.75 SIRT1 (0.61) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL8534092 0.74 ALDH1A1 (0.69) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL8529733 0.74 MEN1 (0.54) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL8530163 0.74 ALDH1A1 (0.54) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL11473183 0.74 AR (0.44) MAPTMEN1KMT2ASLC6A4AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0859757-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS Farmak A.S. (CZ) 1998-08-26 EP disclosed
WO-1997017325-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS FARMAK A.S. (CZ) 1997-05-15 WO disclosed