SCHEMBL8533456

SCHEMBL8533456

Cc1c(-c2ccc(Br)cc2)[nH]c2ccccc2c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.52
HTT P42858 3/20 0.48
HPGD P15428 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
GLA P06280 1/20 0.48
GAA P10253 1/20 0.48
ATM Q13315 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
KIF11 P52732 4/20 0.47
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
POLB P06746 1/20 0.45
KMT2A Q03164 1/20 0.45
MAPT P10636 1/20 0.44
NR1I3 Q14994 1/20 0.44
DAO P14920 1/20 0.42
DDO Q99489 1/20 0.42
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5306250 0.86 CYP11B1 (0.54) PTGS2ALDH1A1KIF11MAPTNR1I3
SCHEMBL9607489 0.84 HTT (0.48) PTGS2HTTHPGDKDM4EALDH1A1
SCHEMBL9607173 0.82 CYP11B1 (0.48) HTTHPGDKDM4EALDH1A1LMNA
SCHEMBL26724947 0.81 KIF11 (0.47) HTTHPGDKDM4EALDH1A1LMNA
SCHEMBL21024209 0.81 PDE10A (0.47) HTTHPGDKDM4EALDH1A1LMNA
SCHEMBL8533400 0.80 KIF11 (0.47) HTTHPGDKDM4EALDH1A1LMNA
SCHEMBL16585681 0.79 CTSV (0.57) LMNAGAAKIF11MEN1KMT2A
SCHEMBL8533957 0.79 PDE10A (0.51) HTTHPGDKDM4EALDH1A1LMNA
SCHEMBL8515205 0.77 SLC2A1 (0.52) PTGS2HTTHPGDKDM4EALDH1A1
SCHEMBL8532778 0.77 PTGS2 (0.46) PTGS2HTTKDM4EALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO claimed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed