SCHEMBL8533461

SCHEMBL8533461

Cc1c(-c2ccc(Cc3ccc(OC(F)(F)F)cc3)cc2)[nH]c2cc(F)ccc2c1=O

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 1/20 0.56
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 1/20 0.41
ESR1 P03372 2/20 0.41
CYP19A1 P11511 3/20 0.40
SLC2A1 P11166 1/20 0.39
KIF11 P52732 1/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPK1 P28482 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
GAA P10253 1/20 0.36
MAPK13 O15264 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
PARP1 P09874 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8515688 0.88 MAT2A (0.55) MAT2AESR1KIF11KDM4E
SCHEMBL8535303 0.88 MAT2A (0.55) MAT2ACYP19A1KIF11PTGDR2
SCHEMBL20983232 0.88 MAT2A (0.55) MAT2AALDH1A1ESR1KIF11KDM4E
SCHEMBL8538462 0.88 MAT2A (0.52) MAT2AESR1KIF11MAPK1
SCHEMBL8532964 0.87 MAT2A (0.52) MAT2AKMT2AESR1KIF11
SCHEMBL8532528 0.85 MAT2A (0.48) MAT2AKIF11
SCHEMBL8535293 0.85 MAT2A (0.48) MAT2AESR1KIF11
SCHEMBL8536444 0.83 MAT2A (0.64) MAT2AMEN1KMT2AALDH1A1CYP19A1
SCHEMBL20983234 0.83 MAT2A (0.58) MAT2AALDH1A1ESR1KDM4E
SCHEMBL8653277 0.83 MAT2A (0.49) MAT2ACYP19A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO claimed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed