SCHEMBL8653277

SCHEMBL8653277

Cc1c(-c2cnn(Cc3ccc(OC(F)(F)F)cc3)c2)[nH]c2cc(F)ccc2c1=O

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 1/20 0.49
CREBBP Q92793 1/20 0.43
CYP19A1 P11511 4/20 0.41
KLKB1 P03952 2/20 0.40
ALK Q9UM73 1/20 0.38
KCNH2 Q12809 2/20 0.38
TYMS P04818 1/20 0.38
CHRM5 P08912 2/20 0.38
ADORA2B P29275 2/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
MAPK1 P28482 1/20 0.38
ABL1 P00519 1/20 0.37
BCR P11274 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8537370 0.93 MAT2A (0.43) MAT2ACREBBPKLKB1ALKKCNH2
SCHEMBL8538579 0.91 MAT2A (0.61) MAT2ACREBBPCYP19A1KLKB1KCNH2
SCHEMBL8533234 0.91 MAT2A (0.49) MAT2ACREBBPCYP19A1KLKB1KCNH2
SCHEMBL8513871 0.89 MAT2A (0.46) MAT2ACREBBPKLKB1KCNH2TYMS
SCHEMBL8536502 0.85 MAT2A (0.43) MAT2ACREBBPKLKB1KCNH2TYMS
SCHEMBL8533461 0.83 MAT2A (0.56) MAT2ACYP19A1MAPK1
SCHEMBL19002091 0.80 MAT2A (0.44) MAT2AKCNH2CHRM5ADORA2BADORA2A
SCHEMBL8536444 0.79 MAT2A (0.64) MAT2ACYP19A1KCNH2MAPK1
SCHEMBL8535741 0.78 ABL1 (0.41) CREBBPKLKB1KCNH2CHRM5ADORA2B
SCHEMBL8531391 0.78 CREBBP (0.40) CREBBPKLKB1KCNH2CHRM5ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO claimed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed