SCHEMBL8533523

SCHEMBL8533523

O=C(Cl)c1ccccc1Sc1ccc(F)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
ALOX15 P16050 1/20 0.49
RHEB Q15382 3/20 0.48
SIRT1 Q96EB6 1/20 0.42
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37
HPGD P15428 1/20 0.37
GRM5 P41594 1/20 0.35
TERT O14746 1/20 0.35
CES2 O00748 2/20 0.35
CES1 P23141 2/20 0.35
TP53 P04637 1/20 0.35
LMNA P02545 1/20 0.35
BLM P54132 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NOD2 Q9HC29 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL234760 0.86 RHEB (0.52) ALDH1A1ALOX15RHEBSIRT1MAPT
SCHEMBL11476180 0.78 SIRT1 (0.67) ALDH1A1ALOX15SIRT1MEN1MAPT
SCHEMBL9815789 0.77 ALDH1A1 (0.52) ALDH1A1ALOX15SIRT1MEN1MAPT
SCHEMBL11473506 0.76 PTPRG (0.48) ALDH1A1RHEBSIRT1MAPTHPGD
SCHEMBL8533398 0.76 SIRT1 (0.50) ALDH1A1ALOX15SIRT1CHRM2CHRM1
SCHEMBL8531894 0.75 SIRT1 (0.46) ALDH1A1ALOX15SIRT1MEN1MAPT
SCHEMBL8529802 0.75 SLC6A2 (0.48) ALDH1A1ALOX15SIRT1MAPTCES2
SCHEMBL28016940 0.75 RHEB (0.43) ALDH1A1ALOX15RHEBMEN1MAPT
SCHEMBL8609339 0.75 SLC6A2 (0.51) ALDH1A1SIRT1MAPTCES2LMNA
SCHEMBL11485914 0.73 CYP2C9 (0.62) RHEBHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0859757-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS Farmak A.S. (CZ) 1998-08-26 EP disclosed
WO-1997017325-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS FARMAK A.S. (CZ) 1997-05-15 WO disclosed