SCHEMBL8533398

SCHEMBL8533398

CSc1ccc(Sc2ccccc2C(=O)Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 1/20 0.50
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
CHRM2 P08172 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
ALDH1A1 P00352 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
ALOX15 P16050 1/20 0.40
LMNA P02545 4/20 0.40
KDM4E B2RXH2 3/20 0.40
MAPT P10636 3/20 0.40
RAB9A P51151 3/20 0.40
NSD2 O96028 1/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
NPC1 O15118 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11476180 0.85 SIRT1 (0.67) SIRT1ALDH1A1L3MBTL1ALOX15LMNA
SCHEMBL8531499 0.84 SIRT1 (0.56) SIRT1SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL3440670 0.81 HTT (0.51) ALDH1A1L3MBTL1ALOX15LMNAMAPT
SCHEMBL9815789 0.81 ALDH1A1 (0.52) SIRT1SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8529733 0.80 MEN1 (0.54) SIRT1SLC6A2SLC6A4SLC6A3CHRM2
SCHEMBL28304795 0.80 SIRT1 (0.51) SIRT1SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8610734 0.79 HPGD (0.44) CHRM2CHRM1CHRM3ALDH1A1L3MBTL1
SCHEMBL21679514 0.79 SIRT1 (0.54) SIRT1SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8529802 0.79 SLC6A2 (0.48) SIRT1SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL13240454 0.78 LMNA (0.62) SIRT1ALDH1A1LMNAMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0859757-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS Farmak A.S. (CZ) 1998-08-26 EP disclosed
WO-1997017325-A1 DERIVATES OF N,N-DIMETHYL-2-(ARYLTHIO)BENZYLAMINE, THEIR SALTS, METHODS OF PREPARATION AND THEIR USE IN PHARMACEUTICAL MEDICAMENTS FARMAK A.S. (CZ) 1997-05-15 WO disclosed