SCHEMBL8533711

SCHEMBL8533711

O=C=CN1C(=O)C(N2C(=O)c3ccccc3C2=O)N=C(C2CCCC2)c2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 14/20 0.36
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
MC4R P32245 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CCKAR P32238 2/20 0.32
TRPA1 O75762 2/20 0.31
BDKRB1 P46663 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8532888 0.79 BDKRB1 (0.39) CCKBRALDH1A1MAPTPKMHPGD
SCHEMBL8773971 0.74 CCKBR (0.45) CCKBRALDH1A1CCKARTRPA1BDKRB1
SCHEMBL8773965 0.74 CCKBR (0.45) CCKBRALDH1A1CCKARTRPA1BDKRB1
SCHEMBL8537963 0.72 ALDH1A1 (0.48) CCKBRALDH1A1PKMHSD17B10CCKAR
SCHEMBL8537959 0.72 ALDH1A1 (0.48) CCKBRALDH1A1PKMHSD17B10CCKAR
SCHEMBL8773950 0.70 CCKBR (0.42) CCKBRALDH1A1HSD17B10CCKARTRPA1
SCHEMBL8536369 0.69 ALDH1A1 (0.42) CCKBRALDH1A1MAPTPKMHPGD
SCHEMBL8536373 0.69 ALDH1A1 (0.42) CCKBRALDH1A1MAPTPKMHPGD
SCHEMBL8537982 0.68 ALDH1A1 (0.41) CCKBRALDH1A1MAPTPKMHPGD
SCHEMBL8537988 0.68 ALDH1A1 (0.41) CCKBRALDH1A1MAPTPKMHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763437-A Benzodiazepine derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-06-09 US disclosed