SCHEMBL8533863

SCHEMBL8533863

c1ccc(C2NCCO2)nc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.39
ADRA1A P35348 1/20 0.39
HTR2B P41595 1/20 0.39
SLC6A3 Q01959 1/20 0.39
ALDH1A1 P00352 4/20 0.37
CTH P32929 1/20 0.37
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
GSK3B P49841 1/20 0.37
MAPT P10636 3/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
NISCH Q9Y2I1 1/20 0.36
KDM4E B2RXH2 2/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
POLB P06746 1/20 0.35
CCR1 P32246 1/20 0.35
CCR5 P51681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Thiophene SCHEMBL28105989 0.91 CTH (0.35) SLC6A2ADRA1AHTR2BSLC6A3ALDH1A1
SCHEMBL8371674 0.79 ALDH1A1 (0.40) SLC6A2ADRA1AHTR2BSLC6A3ALDH1A1
SCHEMBL27512628 0.77 ALDH1A1 (0.38) SLC6A2ADRA1AHTR2BSLC6A3ALDH1A1
SCHEMBL5314101 0.76 CTH (0.42) ALDH1A1CTHDDB1CRBNGSK3B
SCHEMBL10673715 0.73 CYP1A2 (0.41) SLC6A2ADRA1AHTR2BSLC6A3ALDH1A1
SCHEMBL218212 0.72 SLC6A2 (0.46) SLC6A2ADRA1AHTR2BSLC6A3ALDH1A1
SCHEMBL356657 0.72
SCHEMBL30711689 0.72 DRD2 (0.45)
SCHEMBL15949228 0.72 CSNK1D (0.44) SLC6A2ADRA1AHTR2BSLC6A3ALDH1A1
SCHEMBL22325 0.72 DRD2 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1657523-A Cyclic compounds TANABE SEIYAKU CO (JP) 2005-08-24 CN claimed
CN-1440393-A cyclic compound TANABE SEIYAKU CO (JP) 2003-09-03 CN claimed
CN-105814044-B Tetrahydroimidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2018-03-02 CN disclosed
CN-105814045-B Imidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2017-08-25 CN disclosed
CN-104470924-B Imidazopyrazines derivant as TNF active regulator UCB生物制药私人有限公司 2016-11-09 CN disclosed
CN-104619709-B Imidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-11-09 CN disclosed
CN-105829307-A TETRAHYDROIMIDAZOPYRIDINE DERIVATIVES AS MODULATORS OF TNF ACTIVITY UCB生物制药私人有限公司 2016-08-03 CN disclosed
CN-105814044-A Tetrahydroimidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814059-A Imidazopyrimidine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814053-A Imidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814022-A Fused bicyclic heteroaromatic derivatives as modulators of tnf activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814045-A Imidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814060-A Imidazotriazine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814046-A Imidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814025-A Tetrahydrobenzimidazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814051-A Tetrahydroimidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814061-A Imidazopyridazine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-1657523-A Cyclic compounds TANABE SEIYAKU CO (JP) 2005-08-24 CN disclosed
CN-1440393-A cyclic compound TANABE SEIYAKU CO (JP) 2003-09-03 CN disclosed
US-5767279-A Enantiomerically pure pyridylcycloalkylethylamines and the salts thereof and processes for preparing them BOEHRINGER INGELHEIM GMBH (DE) 1998-06-16 US disclosed