SCHEMBL8534192

SCHEMBL8534192

CS(=O)(=O)c1cccc(C(O)C(=CCO)c2ccc(F)cc2)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.41
VNN1 O95497 1/20 0.38
ESR2 Q92731 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
EPHX2 P34913 4/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
AKR1C3 P42330 2/20 0.36
AKR1C2 P52895 1/20 0.36
AKR1C1 Q04828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8423741 0.85 EPHX2 (0.48) PTGS2ESR2EPHX2AKR1C3AKR1C2
SCHEMBL8607731 0.80 CES2 (0.52) PTGS2VNN1ALDH1A1GAAEPHX2
SCHEMBL8607956 0.79 PTGDR2 (0.39) PTGS2VNN1ESR2ALDH1A1GAA
SCHEMBL8423743 0.76 HTR2A (0.40) PTGS2ESR2EPHX2CYP3A4CYP2D6
SCHEMBL14541814 0.69 EPHX2 (0.47) ALDH1A1GAAEPHX2CYP3A4CYP2D6
SCHEMBL19329964 0.69 PTGDR2 (0.43) PTGS2VNN1ALDH1A1GAAEPHX2
SCHEMBL20838412 0.69 PTGDR2 (0.43) PTGS2VNN1ALDH1A1GAAEPHX2
SCHEMBL9895935 0.67 VNN1 (0.45) PTGS2VNN1ALDH1A1GAAEPHX2
SCHEMBL212020 0.67 ALDH1A1 (0.49) ALDH1A1GAACYP3A4CYP2D6SLC6A2
SCHEMBL30661278 0.67 ALDH1A1 (0.49) ALDH1A1GAACYP3A4CYP2D6SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849943-A Stilbene derivatives useful as cyclooxygenase-2 inhibitors MERCK FROSST CANADA, INC. (CA) 1998-12-15 US claimed
US-5736579-A ANTIARTHRITIC, ANTIPYRETIC AND ANALGESIC AGENTS G.D. SEARLE & CO. (US) 1998-04-07 US disclosed
US-5684195-A SULFINIC ACID SALT INTERMEDIATE, OXIDATIVE AMINATION G. D. SEARLE & CO. (US) 1997-11-04 US disclosed
US-5672626-A ANTIINFLAMMATORY AGENT TREATING ARTHRITIS, PAIN, FEVER; ANTIPYRETICS G. D. SEARLE & CO. (US) 1997-09-30 US disclosed
US-5672627-A ANTIINFLAMMATORY AGENT TREATING ARTHRITIS, PAIN, FEVER; ANTIPYRETICS G.D. SEARLE & CO. (US) 1997-09-30 US disclosed
US-5670510-A SELECTIVELY INHIBIT CYCLOOXYGENASE II, ANTIARTHRITIC G. D. SEARLE & CO. (US) 1997-09-23 US disclosed