SCHEMBL8423743

SCHEMBL8423743

CS(=O)(=O)c1ccccc1C(O)C(=CCO)c1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
KCNH2 Q12809 2/20 0.40
PTGS2 P35354 4/20 0.37
CYP2D6 P10635 2/20 0.36
CYP3A4 P08684 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
ESR2 Q92731 2/20 0.34
HSD11B1 P28845 2/20 0.33
AKR1C2 P52895 1/20 0.32
AKR1C1 Q04828 1/20 0.32
AKR1C3 P42330 1/20 0.32
EPHX2 P34913 2/20 0.32
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6026294 0.79 HTR2A (0.42) HTR2AHTR2CKCNH2PTGS2HSD11B1
SCHEMBL8423741 0.77 EPHX2 (0.48) PTGS2ESR2AKR1C2AKR1C1AKR1C3
SCHEMBL8534192 0.76 PTGS2 (0.41) PTGS2CYP2D6CYP3A4SLC6A2SLC6A4
SCHEMBL7846563 0.69 HTR2A (0.39) HTR2AHTR2CKCNH2PTGS2HSD11B1
SCHEMBL16316789 0.66 CYP3A4 (0.43) HTR2AHTR2CKCNH2CYP2D6CYP3A4
SCHEMBL8388365 0.65 ESR2 (0.44) PTGS2ESR2HSD11B1MAPT
SCHEMBL28748849 0.65 HTR2A (0.49) HTR2AHTR2CKCNH2CYP2D6CYP3A4
SCHEMBL28019207 0.64 CYP3A4 (0.40) HTR2AHTR2CKCNH2CYP2D6CYP3A4
SCHEMBL27991976 0.64 LMNA (0.44) HTR2AHTR2CKCNH2CYP2D6CYP3A4
SCHEMBL7083981 0.63 MMP1 (0.48) PTGS2HSD11B1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0788476-B1 STILBENE DERIVATIVES USEFUL AS CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA INC (CA) 1999-10-20 EP claimed