SCHEMBL8534210

SCHEMBL8534210

O=C(NC1CCNCC1)c1ccc(-n2ccnc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.56
HTR2C P28335 1/20 0.56
HTR2B P41595 1/20 0.56
MAPT P10636 2/20 0.56
RAB9A P51151 1/20 0.56
KMT2A Q03164 1/20 0.54
CYP3A4 P08684 1/20 0.51
BAZ2B Q9UIF8 1/20 0.51
HTT P42858 1/20 0.51
CD38 P28907 5/20 0.51
ADH5 P11766 1/20 0.49
ADRB1 P08588 1/20 0.48
CYP4Z1 Q86W10 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
TAOK1 Q7L7X3 1/20 0.47
TAOK3 Q9H2K8 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26401026 0.87 KMT2A (0.71) HTR2AHTR2CHTR2BMAPTRAB9A
SCHEMBL25135518 0.86 KHK (0.50) HTR2AHTR2CHTR2BRAB9ACD38
Hydrochloric Acid SCHEMBL30363722 0.85 KHK (0.49) RAB9ACD38CYP4Z1KHKSMYD3
SCHEMBL25135722 0.81 CD38 (0.49) CD38KHKSMYD3
SCHEMBL30363752 0.81 CD38 (0.49) CD38KHKSMYD3
Hydrochloric Acid SCHEMBL30363726 0.80 CD38 (0.48) CD38KHKSMYD3
SCHEMBL25135519 0.79 CD38 (0.53) HTR2AHTR2CHTR2BCD38CYP4Z1
Hydrochloric Acid SCHEMBL30363847 0.78 CD38 (0.52) HTR2AHTR2CHTR2BCD38CYP4Z1
SCHEMBL29050693 0.78 L3MBTL1 (0.54) L3MBTL1HDAC3HDAC4HDAC1HDAC7
SCHEMBL8537662 0.78 LMNA (0.64) KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0537201-B1 1-[4-(IMIDAZOL-1-YL)BENZOYL]PIPERIDINE DERIVATIVES AS ANTIARRHYTHMIC AGENTS SCHERING AG (DE) 1998-11-18 EP disclosed
EP-0537201-A1 IMIDAZOLYLBENZOYL SUBSTITUTED HETEROCYCLES SCHERING AKTIENGESELLSCHAFT (DE) 1993-04-21 EP disclosed
US-5189036-A Cardiovascular agents; class III antiarrhythmic agents SCHERING AG (DE) 1993-02-23 US disclosed
WO-1991019709-A1 IMIDAZOLYLBENZOYL SUBSTITUTED HETEROCYCLES SCHERING AKTIENGESELLSCHAFT BERLIN UND BERGKAMEN (DE) 1991-12-26 WO disclosed