SCHEMBL8534846

SCHEMBL8534846

Cc1c(-c2ccc(-c3ccc(F)cc3F)cc2)[nH]c2ccccc2c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 2/20 0.50
GLA P06280 1/20 0.50
GAA P10253 1/20 0.50
HTT P42858 1/20 0.50
KIF11 P52732 4/20 0.46
PDE10A Q9Y233 2/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
THRB P10828 1/20 0.44
HPGD P15428 1/20 0.44
CTSV O60911 1/20 0.44
CTSL P07711 1/20 0.44
MAPT P10636 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
PTGS2 P35354 2/20 0.41
NPC1 O15118 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8533957 0.87 PDE10A (0.51) ALDH1A1KDM4EGLAGAAHTT
SCHEMBL8536900 0.86 ALDH1A1 (0.44) ALDH1A1KDM4EGLAGAAHTT
SCHEMBL8532778 0.79 PTGS2 (0.46) ALDH1A1KDM4EGLAGAAHTT
SCHEMBL21024209 0.78 PDE10A (0.47) ALDH1A1KDM4EGLAGAAHTT
SCHEMBL8536439 0.75 PDE10A (0.54) ALDH1A1KDM4EGLAGAAHTT
SCHEMBL9607489 0.75 HTT (0.48) ALDH1A1KDM4EGLAGAAHTT
SCHEMBL8533456 0.75 PTGS2 (0.52) ALDH1A1KDM4EGLAGAAHTT
SCHEMBL8638407 0.74 SCD (0.45) ALDH1A1KDM4EGLAGAAHTT
SCHEMBL695242 0.74 MAPK14 (0.55) KDM4EGAAMEN1KMT2ACTSV
SCHEMBL26724947 0.72 KIF11 (0.47) ALDH1A1KDM4EGLAGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO claimed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed