SCHEMBL8534849

SCHEMBL8534849

O=c1oc(OCc2cccnc2)c(NCC2CC2)c(O)c1CC1CCCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR132 Q9UNW8 1/20 0.38
VKORC1 Q9BQB6 1/20 0.37
KCNH2 Q12809 1/20 0.37
ATM Q13315 1/20 0.37
ATR Q13535 1/20 0.37
LMNA P02545 1/20 0.37
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
GRIN2B Q13224 2/20 0.36
NAMPT P43490 1/20 0.36
NCOA1 Q15788 1/20 0.36
NCOA3 Q9Y6Q9 1/20 0.36
KDM4C Q9H3R0 2/20 0.35
ALDH1A1 P00352 2/20 0.35
PKM P14618 2/20 0.35
ASPH Q12797 1/20 0.34
KDM8 Q8N371 1/20 0.34
CSF1R P07333 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8536081 0.70 GABRA1 (0.40) GPR132VKORC1LMNACYP3A4CYP2D6
SCHEMBL8534845 0.70 CHRM2 (0.37) GPR132VKORC1LMNACHRM2CHRM1
SCHEMBL7373615 0.66 GPR132 (0.39) GPR132LMNANAMPTALDH1A1PKM
SCHEMBL7457650 0.65 GPR132 (0.40) GPR132ATMALDH1A1PKMCSF1R
SCHEMBL7457663 0.65 GPR132 (0.40) GPR132LMNAALDH1A1PKMCSF1R
SCHEMBL27686945 0.64 KDM4E (0.56) CYP2D6ALDH1A1PKMKDM4ECHRM2
SCHEMBL9037973 0.64 LMNA (0.39) GPR132LMNANCOA1NCOA3ALDH1A1
SCHEMBL8911540 0.63 KDM4E (0.54) CYP2D6ALDH1A1PKMKDM4E
SCHEMBL1565525 0.62 CYP1A2 (0.61) LMNACYP2D6NAMPTNCOA1NCOA3
SCHEMBL31054426 0.61 CHRNA7 (0.53) CYP2D6ALDH1A1PKMKDM4ECHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5808062-A AIDS THERAPY WARNER-LAMBERT COMPANY (US) 1998-09-15 US claimed
US-5808062-A AIDS THERAPY WARNER-LAMBERT COMPANY (US) 1998-09-15 US disclosed