SCHEMBL8535783

SCHEMBL8535783

O=C1CN(c2ccc(OCC(F)(F)C(F)F)cc2)C(=O)CN1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
HTT P42858 2/20 0.40
KMT2A Q03164 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ACACB O00763 1/20 0.37
MMP13 P45452 1/20 0.37
MMP14 P50281 1/20 0.37
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
RECQL P46063 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
LIPE Q05469 9/20 0.35
TSHR P16473 2/20 0.33
MAPK1 P28482 1/20 0.33
MAPT P10636 2/20 0.32
USP2 O75604 1/20 0.32
UGCG Q16739 1/20 0.32
NPC1 O15118 1/20 0.32
TP53 P04637 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540845 0.82 ALDH1A1 (0.44) ALDH1A1KMT2AMMP13MMP14MEN1
SCHEMBL8542504 0.79 HTT (0.42) ALDH1A1HTTKMT2ASMN1; SMN2ACACB
SCHEMBL3401516 0.78 ALDH1A1 (0.46) ALDH1A1KMT2AMEN1POLBLIPE
SCHEMBL8536210 0.76 HTT (0.40) ALDH1A1HTTKMT2ASMN1; SMN2ACACB
SCHEMBL8579037 0.72 HTT (0.41) ALDH1A1HTTKMT2ASMN1; SMN2ACACB
SCHEMBL8718627 0.70 HTT (0.41) ALDH1A1HTTKMT2ASMN1; SMN2ACACB
SCHEMBL6647622 0.69 ADRB1 (0.50) ALDH1A1HTTKMT2ASMN1; SMN2ACACB
SCHEMBL6647628 0.69 ADRB1 (0.50) ALDH1A1HTTKMT2ASMN1; SMN2ACACB
SCHEMBL6174527 0.68 HTT (0.46) ALDH1A1HTTKMT2ASMN1; SMN2ACACB
SCHEMBL7687627 0.68 HTT (0.39) ALDH1A1HTTKMT2ASMN1; SMN2ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792780-A FUNGICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-08-11 US disclosed
EP-0657449-B1 Azole compounds, their production and use as antifungal agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-04-08 EP disclosed
US-5545652-A Triazole and imidazole compounds and their use as antifungal therapeutic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-08-13 US disclosed
EP-0657449-A1 Azole compounds, their production and use as antifungal agents Takeda Chemical Industries, Ltd. (JP) 1995-06-14 EP disclosed