SCHEMBL8540845

SCHEMBL8540845

O=C1CN(c2ccc(OC(F)(F)C(F)F)cc2)C(=O)CN1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
TRPV1 Q8NER1 2/20 0.35
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
OPRL1 P41146 1/20 0.33
GAA P10253 1/20 0.33
PPARD Q03181 1/20 0.33
PPARA Q07869 1/20 0.33
MMP13 P45452 1/20 0.32
MMP14 P50281 1/20 0.32
KCNH2 Q12809 1/20 0.32
LIPE Q05469 4/20 0.32
PIM1 P11309 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
POLB P06746 2/20 0.32
AR P10275 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HCRTR1 O43613 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401516 0.87 ALDH1A1 (0.46) ALDH1A1OPRL1PPARDPPARALIPE
SCHEMBL8535783 0.82 ALDH1A1 (0.48) ALDH1A1MMP13MMP14LIPEPOLB
SCHEMBL8584198 0.76 LIPE (0.39) ALDH1A1TRPV1SCN5ASCN9AMMP13
SCHEMBL8538552 0.73 SCN5A (0.38) ALDH1A1TRPV1SCN5ASCN9AMMP13
SCHEMBL4713959 0.71 ALDH1A1 (0.48) ALDH1A1GAAPOLBMEN1KMT2A
SCHEMBL10497873 0.69 SCN5A (0.46) SCN5ASCN9AHCRTR1HCRTR2
SCHEMBL8584196 0.69 SCN5A (0.39) ALDH1A1TRPV1SCN5ASCN9AMMP13
SCHEMBL19410377 0.69 POLB (0.43) ALDH1A1TRPV1PPARDPPARAMMP13
SCHEMBL6177616 0.68 LIPE (0.46) OPRL1LIPEPIM1PIM2POLB
SCHEMBL1907911 0.68 ALDH1A1 (0.48) ALDH1A1TRPV1SCN9APIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792780-A FUNGICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-08-11 US disclosed
EP-0657449-B1 Azole compounds, their production and use as antifungal agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-04-08 EP disclosed
US-5545652-A Triazole and imidazole compounds and their use as antifungal therapeutic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-08-13 US disclosed
EP-0657449-A1 Azole compounds, their production and use as antifungal agents Takeda Chemical Industries, Ltd. (JP) 1995-06-14 EP disclosed