SCHEMBL8536210

SCHEMBL8536210

O=C1NCCN(c2ccc(OCC(F)(F)C(F)F)cc2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 1/20 0.39
ACACB O00763 1/20 0.39
MMP13 P45452 1/20 0.39
MMP14 P50281 1/20 0.39
GRM5 P41594 4/20 0.36
GRM3 Q14832 1/20 0.36
UGCG Q16739 1/20 0.36
LIPE Q05469 11/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8542504 0.89 HTT (0.42) HTTKMT2ASMN1; SMN2ALDH1A1ACACB
SCHEMBL8538552 0.82 SCN5A (0.38) ALDH1A1MMP13MMP14LIPE
SCHEMBL8674229 0.77 PDK2 (0.35) ACACBLIPE
SCHEMBL8535783 0.76 ALDH1A1 (0.48) HTTKMT2ASMN1; SMN2ALDH1A1ACACB
SCHEMBL8579037 0.75 HTT (0.41) HTTKMT2ASMN1; SMN2ALDH1A1ACACB
SCHEMBL8581320 0.75 LIPE (0.46) UGCGLIPE
SCHEMBL6647628 0.74 ADRB1 (0.50) HTTKMT2ASMN1; SMN2ALDH1A1ACACB
SCHEMBL6647622 0.74 ADRB1 (0.50) HTTKMT2ASMN1; SMN2ALDH1A1ACACB
SCHEMBL8581221 0.73 MMP13 (0.39) MMP13MMP14LIPE
SCHEMBL6647626 0.70 HTT (0.39) HTTKMT2ASMN1; SMN2ALDH1A1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792780-A FUNGICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-08-11 US disclosed
EP-0657449-B1 Azole compounds, their production and use as antifungal agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-04-08 EP disclosed
US-5545652-A Triazole and imidazole compounds and their use as antifungal therapeutic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-08-13 US disclosed
EP-0657449-A1 Azole compounds, their production and use as antifungal agents Takeda Chemical Industries, Ltd. (JP) 1995-06-14 EP disclosed