SCHEMBL8536127

SCHEMBL8536127

N=C(N)Nc1cccc(S(=O)(=O)C(Cc2c(F)c(F)c(-c3ccccc3N)c(F)c2F)C(=O)O)c1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA1 P00915 12/20 0.35
CA2 P00918 12/20 0.35
CA9 Q16790 9/20 0.35
CA12 O43570 8/20 0.35
MAPT P10636 1/20 0.35
CASR P41180 2/20 0.34
F2 P00734 1/20 0.33
TMPRSS6 Q8IU80 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8532203 0.75 CA1 (0.36) CA1CA2CA9CA12MAPT
SCHEMBL8531517 0.71 ITGB3 (0.35) CA1CA2CA9CA12MAPT
SCHEMBL8536201 0.70 ITGB3 (0.35) CA1CA2CA9CA12MAPT
Propionic Acid SCHEMBL8534857 0.66 USP28 (0.40) CA1CA2CA9CA12MAPT
SCHEMBL8499992 0.65 MEN1 (0.42) CA1CA2MAPTF2
SCHEMBL8697020 0.64 CA1 (0.37) CA1CA2CA9CA12MAPT
SCHEMBL1593097 0.63 CA1 (0.64) CA1CA2CA9CA12MAPT
SCHEMBL8372024 0.62 POLB (0.54) F2TMPRSS6
SCHEMBL7372864 0.62 KMT2A (0.57) CA1CA2CA9CA12MAPT
SCHEMBL2833035 0.62 ITGB3 (0.48) CA1CA2CA9MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773646-A INTEGRIN INHIBITORS G. D. SEARLE & CO. (US) 1998-06-30 US disclosed