SCHEMBL8536153

SCHEMBL8536153

CC(C)[C@H](NC(=O)CCCCCCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)[C@@H](O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)CCCCCCCCCCCN)C(C)C

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSD P07339 9/20 0.55
CA2 P00918 1/20 0.53
MMP2 P08253 1/20 0.51
REN P00797 1/20 0.46
PSMB5 P28074 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8536393 0.94 CTSD (0.52) CTSDCA2MMP2REN
SCHEMBL7345648 0.84 CA2 (0.54) CTSDCA2
Hydrochloric Acid SCHEMBL8535408 0.84 MMP2 (0.53) CTSDCA2MMP2
SCHEMBL7268478 0.83 CTSD (0.54) CTSD
SCHEMBL623353 0.83 CTSD (0.52) CTSD
SCHEMBL623404 0.83 CTSD (0.52) CTSD
SCHEMBL7332623 0.82 CA2 (0.57) CTSDCA2
SCHEMBL7275501 0.81 MMP2 (0.50) MMP2
SCHEMBL621676 0.80 CTSD (0.50) CTSDREN
SCHEMBL7333197 0.80 CA2 (0.54) CTSDCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712417-A Inhibitors of retroviral proteases ABBOTT LABORATORIES (US) 1998-01-27 US disclosed
EP-0428849-A2 Retroviral protease inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1991-05-29 EP disclosed