SCHEMBL8536225

SCHEMBL8536225

CCc1c(CCC(=O)OCNC=O)cccc1-c1cccc(C#N)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.40
S1PR1 P21453 9/20 0.40
CYP2C9 P11712 3/20 0.40
USP7 Q93009 2/20 0.39
CYP2D6 P10635 2/20 0.37
CHRM3 P20309 1/20 0.36
CNR2 P34972 1/20 0.36
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
HCAR2 Q8TDS4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8433145 0.85 EGLN1 (0.39) USP7CNR2PDCD1CD274
SCHEMBL8532684 0.80 ENPP2 (0.35) S1PR1CYP2C9ALDH1A1GAA
SCHEMBL10980808 0.68 ADRA2C (0.68) ADRA2CUSP7CYP2D6CNR2PTGDR2
SCHEMBL6166508 0.68 ADRA2C (0.56) ADRA2CCYP2D6CHRM3ALDH1A1PTGDR2
SCHEMBL19209427 0.67 PPARG (0.44) ADRA2CCYP2D6CNR2PDCD1CD274
SCHEMBL5426031 0.67 PTGDR2 (0.55) ADRA2CALDH1A1PTGDR2
SCHEMBL8432620 0.67 F10 (0.38)
SCHEMBL9357799 0.65 CYP4F2 (0.62) PDCD1CD274ALDH1A1GAA
SCHEMBL19209418 0.64 PPARG (0.44) CYP2C9CYP2D6CNR2PDCD1CD274
SCHEMBL12648685 0.63 CYP11B2 (0.44) ADRA2CS1PR1CYP2C9USP7CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773646-A INTEGRIN INHIBITORS G. D. SEARLE & CO. (US) 1998-06-30 US disclosed