SCHEMBL8536240

SCHEMBL8536240

CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccccc1)CS(=O)(=O)CC(Cc1ccccc1)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.58
CA2 P00918 1/20 0.55
CA5A P35218 1/20 0.55
CTSD P07339 2/20 0.55
CTRB1 P17538 2/20 0.54
CA1 P00915 1/20 0.53
CTSL P07711 5/20 0.52
CTSK P43235 4/20 0.52
CTSS P25774 2/20 0.50
ECE1 P42892 2/20 0.50
CTSB P07858 2/20 0.50
MME P08473 1/20 0.50
CASP7 P55210 1/20 0.49
CYP3A4 P08684 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7323342 0.87 CYP3A4 (0.60) CASP3CA2CA5ACTSDCTRB1
SCHEMBL10084557 0.83 CYP3A4 (0.55) CASP3CA2CA5ACTSDCTRB1
SCHEMBL19557810 0.81 CASP3 (0.61) CASP3CA2CA5ACTSDCA1
SCHEMBL10453618 0.81 CASP3 (0.61) CASP3CA2CA5ACTSDCA1
SCHEMBL7310487 0.81 CTSD (0.62) CASP3CA2CTSDCTRB1CTSL
SCHEMBL25287172 0.81 ECE1 (0.61) CASP3CTSDCTSLCTSKCTSS
SCHEMBL3058668 0.81 ECE1 (0.61) CASP3CTSDCTSLCTSKCTSS
SCHEMBL7269151 0.81 ALDH1A1 (0.60) CASP3CA2CA5ACTSDCTSL
SCHEMBL30601624 0.81 CYP3A4 (0.55) CTSDCTRB1CTSLCTSKECE1
SCHEMBL623817 0.81 CTSD (0.53) CASP3CA2CA5ACTSDCTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed