SCHEMBL8536346

SCHEMBL8536346

CC(C)[C@H](N)C(=O)N[C@H](C(=O)N(C(=O)CCCCCN)C(Cc1ccccc1)C(O)C(Cc1ccccc1)N(C(=O)CCCCC(=O)O)C(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)C(C)C)C(C)C

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.40
F2 P00734 2/20 0.39
PLG P00747 1/20 0.38
LTA4H P09960 1/20 0.38
BACE1 P56817 4/20 0.37
KDM4A O75164 2/20 0.37
KDM4C Q9H3R0 2/20 0.37
MC4R P32245 1/20 0.37
MC5R P33032 1/20 0.37
MC3R P41968 1/20 0.37
CTSD P07339 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8536372 0.87 MMP2 (0.46) MMP2F2LTA4HMC4RMC5R
SCHEMBL8534831 0.86 HTT (0.46) CTSD
SCHEMBL8539750 0.80 CTSD (0.42) BACE1CTSD
SCHEMBL7279627 0.79 PTGER4 (0.41) BACE1CTSD
SCHEMBL9741444 0.75 CTSD (0.37) BACE1CTSD
SCHEMBL8534863 0.75 HTT (0.47)
SCHEMBL8536393 0.74 CTSD (0.52) MMP2BACE1CTSD
SCHEMBL29630664 0.70 BACE1 (0.58) BACE1CTSD
SCHEMBL29496448 0.69 GNPAT (0.53) F2BACE1CTSD
SCHEMBL30385347 0.69 GNPAT (0.53) F2BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed