SCHEMBL8536787

SCHEMBL8536787

NN=CNc1cccc(C(=O)C(N)=C(C(=O)O)c2cccc(Cl)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
KCNK3 O14649 1/20 0.40
KCNK9 Q9NPC2 1/20 0.40
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
MAPT P10636 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
HTT P42858 2/20 0.39
LMNA P02545 2/20 0.39
ERCC5 P28715 1/20 0.39
FEN1 P39748 1/20 0.39
GSK3B P49841 1/20 0.37
CES1 P23141 1/20 0.37
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539554 0.89 CA1 (0.38) PARP1NPC1RAB9AKCNK3KCNK9
SCHEMBL8540372 0.88 KCNK3 (0.37) PARP1NPC1RAB9AKCNK3KCNK9
SCHEMBL8538564 0.86 PARP1 (0.40) PARP1NPC1RAB9AKCNK3KCNK9
SCHEMBL8538094 0.86 CES2 (0.42) PARP1NPC1RAB9AKCNK3KCNK9
SCHEMBL8542528 0.86 SMN1; SMN2 (0.34) PARP1NPC1RAB9AKCNK3KCNK9
SCHEMBL8542364 0.84 CES2 (0.47) PARP1NPC1RAB9AKCNK3KCNK9
SCHEMBL8538807 0.84 KCNK3 (0.42) NPC1RAB9AKCNK3KCNK9MEN1
SCHEMBL8542422 0.84 PARP1 (0.36) PARP1NPC1RAB9AKCNK3KCNK9
SCHEMBL8544139 0.84 KAT6A (0.38) PARP1RAB9AMAPTSMN1; SMN2
SCHEMBL8538385 0.81 KCNK3 (0.43) PARP1NPC1RAB9AKCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852210-A Cinnamic acid derivatives G. D. SEARLE & CO. (US) 1998-12-22 US claimed
US-5852210-A Cinnamic acid derivatives G. D. SEARLE & CO. (US) 1998-12-22 US disclosed