SCHEMBL8536858

SCHEMBL8536858

Cc1cc(O)ccc1-c1ncc[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 9/20 0.46
ESR1 P03372 8/20 0.46
NISCH Q9Y2I1 2/20 0.46
CDK4 P11802 1/20 0.44
CCNA2 P20248 1/20 0.44
CCND1 P24385 1/20 0.44
CDK2 P24941 1/20 0.44
CCND3 P30281 1/20 0.44
JAK2 O60674 1/20 0.44
JAK1 P23458 1/20 0.44
TYK2 P29597 1/20 0.44
JAK3 P52333 1/20 0.44
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
ALOX12 P18054 1/20 0.43
MAPK10 P53779 1/20 0.43
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.43
SMPD3 Q9NY59 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8537911 0.83 AMY1A (0.45) ESR1NISCHCDK4CCNA2CCND1
SCHEMBL31429641 0.81 GUSB (0.45) NISCHCDK4CCNA2CCND1CDK2
SCHEMBL8540911 0.81 GUSB (0.45) NISCHCDK4CCNA2CCND1CDK2
SCHEMBL29466815 0.81 NISCH (0.58) NISCHMEN1ALDH1A1MAPTKMT2A
SCHEMBL4775732 0.81 NISCH (0.58) NISCHMEN1ALDH1A1MAPTKMT2A
SCHEMBL5914842 0.79 ADRA2A (0.49) NISCHMEN1ALDH1A1KMT2ASMPD3
SCHEMBL15152912 0.79 NISCH (0.46) NISCHMTORADKBRD4
SCHEMBL15651168 0.79 NISCH (0.46) NISCHMEN1ALDH1A1MAPTKMT2A
SCHEMBL2455067 0.79 NISCH (0.46) NISCHMEN1ALDH1A1KMT2ASMPD3
SCHEMBL28654223 0.78 NISCH (0.50) NISCHCDK4CCNA2CCND1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed