SCHEMBL8536969

SCHEMBL8536969

C[C@@]12CCC[C@H]1[C@@H]1CC[C@H]3NC(=O)C=C(CCCc4ccccn4)[C@]3(C)[C@H]1CC2

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.34
MBOAT4 Q96T53 3/20 0.33
NAAA Q02083 1/20 0.33
TSHR P16473 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
DDB1 Q16531 1/20 0.30
CRBN Q96SW2 1/20 0.30
SRD5A1 P18405 1/20 0.30
HRH3 Q9Y5N1 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540072 0.84 CYP19A1 (0.32) CYP19A1MBOAT4GRIN1GRIN2BSRD5A1
SCHEMBL8536972 0.80 MBOAT4 (0.39) CYP19A1MBOAT4NAAATSHRGRIN1
SCHEMBL8407144 0.78 CYP19A1 (0.41) CYP19A1MBOAT4GRIN1GRIN2BSRD5A1
SCHEMBL9618179 0.71 SRD5A1 (0.42) CYP19A1MBOAT4GRIN1GRIN2BSRD5A1
SCHEMBL7643432 0.70 CYP19A1 (0.41) CYP19A1MBOAT4GRIN1GRIN2BSRD5A1
SCHEMBL9318599 0.68 CYP19A1 (0.39) CYP19A1MBOAT4GRIN1GRIN2BSRD5A1
SCHEMBL11410578 0.67 CYP19A1 (0.38) CYP19A1MBOAT4GRIN1GRIN2BSRD5A1
SCHEMBL5580929 0.67 CYP19A1 (0.35) CYP19A1MBOAT4GRIN1GRIN2BSRD5A1
SCHEMBL8540073 0.67 MBOAT4 (0.37) CYP19A1MBOAT4GRIN1GRIN2BSRD5A1
SCHEMBL8766060 0.66 SRD5A1 (0.52) SRD5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760045-A BENIGN PROSTATIC HYPERPLASIA MERCK & CO., INC. (US) 1998-06-02 US disclosed
US-5710275-A ENZYME AND HORMONE INHIBITORS MERCK & CO., INC. (US) 1998-01-20 US disclosed
US-5693809-A PREGNANES FOR TREATING ALOPECIA, ACNE AND SKIN DISORDER MERCK & CO., INC. (US) 1997-12-02 US disclosed
US-5510351-A PREGNANE ENZYME INHIBITOR FOR TREATING SKIN DISORDER, BALDNESS, PROSTATIC CANCER MERCK & CO., INC. (US) 1996-04-23 US disclosed