SCHEMBL8536972

SCHEMBL8536972

C[C@@]12CCC[C@H]1[C@@H]1CC[C@H]3NC(=O)C(CCCc4ccccn4)=C[C@]3(C)[C@H]1CC2

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 3/20 0.39
CYP19A1 P11511 4/20 0.32
TSHR P16473 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
NAAA Q02083 1/20 0.32
SRD5A2 P31213 6/20 0.31
SRD5A1 P18405 6/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540073 0.84 MBOAT4 (0.37) MBOAT4CYP19A1GRIN1GRIN2BSRD5A2
SCHEMBL8536969 0.80 CYP19A1 (0.34) MBOAT4CYP19A1TSHRGRIN1GRIN2B
SCHEMBL8823383 0.78 MBOAT4 (0.48) MBOAT4CYP19A1GRIN1GRIN2BSRD5A2
SCHEMBL5109022 0.74 MBOAT4 (0.51) MBOAT4CYP19A1GRIN1GRIN2BSRD5A2
SCHEMBL8016925 0.72 MBOAT4 (0.43) MBOAT4CYP19A1SRD5A2SRD5A1
SCHEMBL9618180 0.72 SRD5A1 (0.44) MBOAT4GRIN1GRIN2BSRD5A2SRD5A1
SCHEMBL9543229 0.70 MBOAT4 (0.41) MBOAT4CYP19A1SRD5A2SRD5A1
SCHEMBL7643438 0.70 MBOAT4 (0.47) MBOAT4CYP19A1GRIN1GRIN2BSRD5A2
SCHEMBL9776615 0.69 SRD5A1 (0.41) MBOAT4SRD5A2SRD5A1
SCHEMBL9708876 0.69 SRD5A1 (0.42) MBOAT4SRD5A2SRD5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760045-A BENIGN PROSTATIC HYPERPLASIA MERCK & CO., INC. (US) 1998-06-02 US disclosed
US-5710275-A ENZYME AND HORMONE INHIBITORS MERCK & CO., INC. (US) 1998-01-20 US disclosed
US-5693809-A PREGNANES FOR TREATING ALOPECIA, ACNE AND SKIN DISORDER MERCK & CO., INC. (US) 1997-12-02 US disclosed
US-5510351-A PREGNANE ENZYME INHIBITOR FOR TREATING SKIN DISORDER, BALDNESS, PROSTATIC CANCER MERCK & CO., INC. (US) 1996-04-23 US disclosed