SCHEMBL8537838

SCHEMBL8537838

N#Cc1ccc(C#Cc2ccc([N+](=O)[O-])o2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 4/20 0.39
VCAM1 P19320 3/20 0.38
KDM4E B2RXH2 4/20 0.37
LMNA P02545 3/20 0.37
MAPT P10636 3/20 0.37
L3MBTL1 Q9Y468 3/20 0.37
NPC1 O15118 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
MITF O75030 1/20 0.37
XBP1 P17861 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PKM P14618 1/20 0.35
KCNJ1 P48048 1/20 0.35
KCNH2 Q12809 1/20 0.35
P2RY6 Q15077 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1608505 0.81 KMT2A (0.44) VCAM1KDM4ELMNAMAPTL3MBTL1
SCHEMBL12039494 0.76 CASP3 (0.44) KDM4ELMNAMAPTL3MBTL1NPSR1
SCHEMBL11731415 0.74 LMNA (0.42) KDM4ELMNAMAPTL3MBTL1NPC1
SCHEMBL27214761 0.73 KCNJ1 (0.55) FBP1VCAM1LMNAMAPTNPC1
SCHEMBL8538325 0.73 KCNJ1 (0.41) KDM4ELMNAMAPTALDH1A1TDP1
SCHEMBL8815587 0.73 MMP2 (0.31)
SCHEMBL1811649 0.71 LMNA (0.46) KDM4ELMNAMAPTL3MBTL1NPC1
SCHEMBL8538501 0.70 LMNA (0.44) KDM4ELMNAMAPTL3MBTL1NPC1
SCHEMBL11848697 0.70 LMNA (0.44) KDM4ELMNAMAPTL3MBTL1NPC1
SCHEMBL6428842 0.68 KMT2A (0.64) KDM4ELMNAMAPTNPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726195-A Aminoacyl adenylate mimics as novel antimicrobial and antiparasitic agents CUBIST PHARMACEUTICALS, INC. (US) 1998-03-10 US disclosed
WO-1997005132-A1 AMINOACYL ADENYLATE MIMICS AS NOVEL ANTIMICROBIAL AND ANTIPARASITIC AGENTS CUBIST PHARMACEUTICALS, INC. (US) 1997-02-13 WO disclosed