SCHEMBL8538325

SCHEMBL8538325

O=[N+]([O-])c1ccc(C#Cc2ccc(-n3cnnn3)cc2)o1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 4/20 0.41
KCNH2 Q12809 2/20 0.41
MAPT P10636 4/20 0.39
NOTUM Q6P988 3/20 0.39
F2 P00734 1/20 0.39
ALDH1A1 P00352 4/20 0.38
LMNA P02545 3/20 0.38
POLB P06746 1/20 0.37
BLM P54132 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HTT P42858 1/20 0.37
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35
HPGD P15428 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8538200 0.73 KCNJ1 (0.41) KCNJ1KCNH2MAPTNOTUMF2
SCHEMBL8537838 0.73 FBP1 (0.39) KCNJ1KCNH2MAPTALDH1A1LMNA
SCHEMBL1269000 0.71 KCNJ1 (0.68) KCNJ1KCNH2MAPTNOTUMF2
SCHEMBL8815587 0.68 MMP2 (0.31)
SCHEMBL12615985 0.66 NOTUM (0.78) KCNJ1MAPTNOTUMF2ALDH1A1
SCHEMBL12039494 0.66 CASP3 (0.44) MAPTALDH1A1LMNACA12CA9
SCHEMBL11731415 0.64 LMNA (0.42) MAPTALDH1A1LMNAPOLBTDP1
SCHEMBL5148009 0.62 LMNA (0.51) KCNJ1KCNH2MAPTNOTUMF2
SCHEMBL8485436 0.62 KCNJ1 (0.66) KCNJ1MAPTNOTUMF2ALDH1A1
SCHEMBL1811649 0.62 LMNA (0.46) MAPTALDH1A1LMNAPOLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726195-A Aminoacyl adenylate mimics as novel antimicrobial and antiparasitic agents CUBIST PHARMACEUTICALS, INC. (US) 1998-03-10 US disclosed