SCHEMBL8538280

SCHEMBL8538280

N#Cc1ccccc1N(CCCl)CCCl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.38
HDAC6 Q9UBN7 1/20 0.34
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 3/20 0.33
HTT P42858 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
ESR2 Q92731 1/20 0.32
EGFR P00533 1/20 0.31
ERBB2 P04626 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20133582 0.81 TSHR (0.42) TSHRHDAC6ALDH1A1KDM4EHTT
SCHEMBL1344312 0.81 ALDH1A1 (0.41) TSHRHDAC6ALDH1A1KDM4EHTT
SCHEMBL8746679 0.78 TSHR (0.42) TSHRHDAC6ALDH1A1KDM4EHTT
SCHEMBL2560142 0.76 TSHR (0.45) TSHRHDAC6ALDH1A1KDM4EHTT
SCHEMBL20157017 0.75 TSHR (0.40) TSHRHDAC6ALDH1A1HTTHPGD
SCHEMBL8773387 0.75 HDAC6 (0.41) TSHRHDAC6ALDH1A1HPGDHSD17B10
SCHEMBL8746684 0.75 HDAC6 (0.41) TSHRHDAC6ALDH1A1HPGDHSD17B10
Hydrochloric Acid SCHEMBL7464995 0.74 KDM4E (0.40) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL29827525 0.72 TSHR (0.48) TSHRALDH1A1KDM4EHTTHPGD
SCHEMBL2565156 0.72 SLC6A2 (0.43) TSHRHDAC6ALDH1A1KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0496222-B1 Indole derivatives MERCK PATENT GMBH (DE) 1998-09-09 EP disclosed
US-5418237-A Indole derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-05-23 US disclosed
EP-0496222-A1 Indole derivatives MERCK PATENT GmbH (DE) 1992-07-29 EP disclosed