SCHEMBL8538740

SCHEMBL8538740

N#Cc1ccc(-c2ncc[nH]2)cc1-c1ncc[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.46
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
MTOR P42345 1/20 0.44
ADK P55263 1/20 0.44
CHEK1 O14757 1/20 0.43
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
F11 P03951 1/20 0.41
KLKB1 P03952 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP19A1 P11511 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3978330 0.83 NISCH (0.45) NISCHPDE4APDE4BPDE4CPDE4D
SCHEMBL8537240 0.83 CYP11B2 (0.48) NISCH
SCHEMBL5012098 0.83 PDE4A (0.44) NISCHPDE4APDE4BPDE4CPDE4D
SCHEMBL28450350 0.81 NISCH (0.57) NISCHPDE4APDE4BPDE4CPDE4D
SCHEMBL7425938 0.79 NISCH (0.45) NISCHPDE4APDE4BPDE4CPDE4D
SCHEMBL2552798 0.79 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DCHEK1
SCHEMBL2651232 0.78 CSNK1A1 (0.49) NISCHPDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL5855000 0.77 CSNK1A1 (0.47) NISCHPDE4APDE4BPDE4CPDE4D
SCHEMBL15568925 0.74 NISCH (0.49) NISCHPDE4APDE4BPDE4CPDE4D
SCHEMBL1239841 0.74 ADRA2A (0.46) NISCHPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed