SCHEMBL8539149

SCHEMBL8539149

C=CCOC(=O)c1ccc2cc([N+](=O)[O-])ccc2n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
MAPT P10636 4/20 0.53
GAA P10253 3/20 0.53
KDM4E B2RXH2 2/20 0.53
POLB P06746 2/20 0.42
TTR P02766 1/20 0.41
LMNA P02545 1/20 0.41
PMP22 Q01453 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CYP3A4 P08684 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 2/20 0.39
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
SLC6A4 P31645 1/20 0.39
THPO P40225 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540920 0.80 ALDH1A1 (0.43) ALDH1A1MAPTGAAKDM4EPOLB
SCHEMBL6965338 0.79 ALDH1A1 (0.53) ALDH1A1MAPTGAAKDM4EPOLB
SCHEMBL8541741 0.76 ALDH1A1 (0.58) ALDH1A1MAPTGAAKDM4ETTR
SCHEMBL5101748 0.75 CYP3A4 (0.57) ALDH1A1KDM4EPOLBCYP3A4RAB9A
SCHEMBL8545179 0.75 ALDH1A1 (0.48) ALDH1A1MAPTGAAKDM4EPOLB
SCHEMBL28006558 0.74 ALDH1A1 (0.50) ALDH1A1MAPTGAAKDM4EPOLB
SCHEMBL8542694 0.73 MEN1 (0.44) ALDH1A1MAPTGAAKDM4EPOLB
SCHEMBL9700739 0.73 KMT2A (0.55) ALDH1A1MAPTKDM4EPOLBCYP3A4
SCHEMBL10492784 0.73 CYP3A4 (0.50) ALDH1A1MAPTGAANPSR1CYP3A4
SCHEMBL11758391 0.73 CYP3A4 (0.50) ALDH1A1POLBCYP3A4KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0581500-B1 Antibiotic carbapenem compounds ZENECA LTD (GB) 1998-09-09 EP disclosed
US-5441949-A Carbapenem antibiotic compounds ZENECA LIMITED (GB) 1995-08-15 US disclosed
EP-0581500-A1 Antibiotic carbapenem compounds ZENECA LIMITED (GB) 1994-02-02 EP disclosed