SCHEMBL8540920

SCHEMBL8540920

C=CCOC(=O)c1ccc2cc(N)ccc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CYP3A4 P08684 1/20 0.42
PLAU P00749 1/20 0.41
KDM4E B2RXH2 4/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
CASP6 P55212 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
MAPT P10636 5/20 0.38
SNCA P37840 1/20 0.37
FGFR1 P11362 1/20 0.36
RHOA P61586 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GAA P10253 1/20 0.36
TTR P02766 1/20 0.35
GABRP O00591 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539149 0.80 ALDH1A1 (0.53) ALDH1A1CYP3A4KDM4ELMNAPOLB
SCHEMBL3364644 0.77 LMNA (0.50) ALDH1A1PLAUKDM4ELMNAPOLB
SCHEMBL8540048 0.75 TSHR (0.52) ALDH1A1TSHRHSD17B10CYP3A4KDM4E
SCHEMBL27364792 0.74 CYP3A4 (0.46) ALDH1A1TSHRHSD17B10CYP3A4KDM4E
SCHEMBL8541555 0.73 ALDH1A1 (0.54) ALDH1A1TSHRHSD17B10CYP3A4PLAU
SCHEMBL6217194 0.73 CYP3A4 (0.59) ALDH1A1TSHRHSD17B10CYP3A4KDM4E
SCHEMBL10465204 0.73 MGAM (0.56) ALDH1A1TSHRHSD17B10CYP3A4PLAU
SCHEMBL8542799 0.73 ALDH1A1 (0.53) ALDH1A1TSHRHSD17B10CYP3A4KDM4E
SCHEMBL5102454 0.72 CYP3A4 (0.64) ALDH1A1TSHRHSD17B10CYP3A4KDM4E
SCHEMBL8539340 0.72 ALDH1A1 (0.52) ALDH1A1TSHRHSD17B10CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0581500-B1 Antibiotic carbapenem compounds ZENECA LTD (GB) 1998-09-09 EP disclosed
US-5441949-A Carbapenem antibiotic compounds ZENECA LIMITED (GB) 1995-08-15 US disclosed
EP-0581500-A1 Antibiotic carbapenem compounds ZENECA LIMITED (GB) 1994-02-02 EP disclosed