SCHEMBL8539432

SCHEMBL8539432

CCCC(C)S(=O)(=O)c1cc(CC)c(C(=O)Cl)cc1[N+](=O)[O-]

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.36
VCAM1 P19320 6/20 0.32
ALOX15 P16050 1/20 0.32
ALOX12 P18054 1/20 0.32
ALDH1A1 P00352 2/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
NPC1 O15118 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8542407 0.90 PDK1 (0.38) PDK1VCAM1ALOX15ALOX12ALDH1A1
SCHEMBL8541696 0.88 PDGFRB (0.34) PDK1VCAM1ALDH1A1GAAHPGD
SCHEMBL8540482 0.88 PDK1 (0.39) PDK1VCAM1ALOX15ALOX12ALDH1A1
SCHEMBL27358004 0.84 PDK1 (0.39) PDK1VCAM1ALOX15ALOX12ALDH1A1
SCHEMBL6934380 0.83 SLC9A1 (0.38)
SCHEMBL8541274 0.81 SLC9A1 (0.31)
SCHEMBL8538668 0.80 PDK1 (0.36) PDK1VCAM1ALDH1A1
SCHEMBL8544973 0.79 PDK1 (0.37) PDK1VCAM1ALDH1A1HPGDCYP3A4
SCHEMBL8544879 0.78 ALDH1A1 (0.37) PDK1VCAM1ALDH1A1GAAHPGD
SCHEMBL8537184 0.78 TXNRD1 (0.39) PDK1VCAM1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1071743-C Sulfuryl or sulfinyl benzoyl guanidine derivative MERCK PATENT GMBH (DE) 2001-09-26 CN disclosed
US-5744641-A Sulfonyl- or sulfinylbenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-28 US disclosed
CN-1148590-A Sulfuryl or sulfinyl benzoyl guanidine derivative MERCK PATENT GMBH (DE) 1997-04-30 CN disclosed